SCHEMBL2977903

SCHEMBL2977903

COC(=O)CCCC(=O)NC1CCC(c2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.45
OPRM1 P35372 3/20 0.44
OPRL1 P41146 2/20 0.44
KCNH2 Q12809 2/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
CYP2B6 P20813 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
PRCP P42785 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GRIN1 Q05586 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
EPHX1 P07099 1/20 0.44
OPRD1 P41143 1/20 0.43
NPY1R P25929 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2985682 0.90 GLA (0.41) EPHX2OPRM1OPRL1EPHX1KCNA3
SCHEMBL2976705 0.85 MEN1 (0.52) EPHX2KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL4046657 0.82 KMT2A (0.53) EPHX2OPRM1OPRL1KCNH2GRIN2D
SCHEMBL4054898 0.78 ACKR3 (0.59) OPRM1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL2981500 0.73 POLB (0.50) OPRM1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL2985381 0.73 OPRM1 (0.48) EPHX2OPRM1OPRL1EPHX1KCNA3
SCHEMBL316418 0.72 HRH3 (0.41) EPHX2OPRM1OPRL1KCNH2GRIN2D
Phencyclidine SCHEMBL28204695 0.70 GRIN1 (0.63) OPRM1OPRL1KCNH2GRIN2DGRIN3B
SCHEMBL2987893 0.70 OPRM1 (0.51) OPRM1OPRL1CYP2C19
SCHEMBL4868037 0.70 HRH2 (0.46) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US claimed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US claimed
US-7786328-B2 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2010-08-31 US disclosed
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-12-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070281954-A1 Cyclohexyl-1,4-diamine compounds DPYD, PKD1, AOC1 EPHX2 1094/4885OPRM1 1483/4885OPRL1 1292/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.