SCHEMBL29784263

SCHEMBL29784263

COC(=O)c1cc(F)cc2cc(CNC(=O)OC(C)(C)C)oc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 3/20 0.42
KDM4A O75164 1/20 0.38
GRM2 Q14416 1/20 0.36
ATR Q13535 1/20 0.36
CACNA1H O95180 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1C Q13936 1/20 0.35
PARP1 P09874 2/20 0.35
PARP2 Q9UGN5 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HIF1A Q16665 1/20 0.34
ERAP1 Q9NZ08 3/20 0.33
EPAS1 Q99814 1/20 0.33
KCNA5 P22460 1/20 0.33
DYRK1A Q13627 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27185757 1.00 STING1 (0.42) STING1KDM4AGRM2ATRCACNA1H
SCHEMBL29784449 0.88 ESR2 (0.40) STING1KDM4AATRCACNA1HCACNA1B
SCHEMBL27185785 0.88 ALDH1A1 (0.40) STING1KDM4AATRCACNA1HCACNA1B
SCHEMBL29784510 0.88 ALDH1A1 (0.40) STING1KDM4AATRCACNA1HCACNA1B
SCHEMBL27185758 0.88 ESR2 (0.40) STING1KDM4AATRCACNA1HCACNA1B
SCHEMBL29784315 0.87 SLC22A12 (0.44) STING1KDM4AATRKDM4EALDH1A1
SCHEMBL29784436 0.87 STING1 (0.38) STING1KDM4AGRM2CACNA1HCACNA1B
SCHEMBL16347843 0.87 STING1 (0.38) STING1KDM4AATRCACNA1HCACNA1B
SCHEMBL29784337 0.87 STING1 (0.43) STING1KDM4AATRALDH1A1GAA
SCHEMBL27185593 0.87 STING1 (0.43) STING1KDM4AATRALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022169921-A1 BENZOFURAN COMPOUNDS AS STING AGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2022-08-11 WO disclosed