SCHEMBL29795366

SCHEMBL29795366

COc1ccc(CNC2CCN(C(=O)OC(C)(C)C)C2)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.63
LMNA P02545 2/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TP53 P04637 3/20 0.53
STS P08842 2/20 0.52
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MMP1 P03956 2/20 0.48
MMP9 P14780 2/20 0.48
EPHX2 P34913 1/20 0.48
MMP3 P08254 1/20 0.48
MMP7 P09237 1/20 0.48
GPR119 Q8TDV5 1/20 0.48
BACE1 P56817 2/20 0.48
CTSD P07339 1/20 0.48
CTSE P14091 1/20 0.48
MMP13 P45452 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381166 0.93 ALDH1A1 (0.69) ALDH1A1LMNAMAPTSMN1; SMN2TP53
SCHEMBL2308747 0.91 ALDH1A1 (0.55) ALDH1A1LMNAMAPTSMN1; SMN2TP53
SCHEMBL8310166 0.90 ALDH1A1 (0.65) ALDH1A1LMNAMAPTSMN1; SMN2TP53
SCHEMBL20794854 0.88 GPR119 (0.52) ALDH1A1MAPTSMN1; SMN2TP53MEN1
SCHEMBL17605157 0.87 DNMT3A (0.52) ALDH1A1MAPTTP53MEN1KMT2A
SCHEMBL651891 0.87 HTT (0.53) ALDH1A1MAPTSMN1; SMN2STSMEN1
SCHEMBL17605155 0.87 DNMT3A (0.52) ALDH1A1MAPTTP53MEN1KMT2A
SCHEMBL652820 0.87 HTT (0.53) ALDH1A1MAPTSMN1; SMN2STSMEN1
SCHEMBL696779 0.87 USP30 (0.56) LMNASTSGPR119BACE1
SCHEMBL696778 0.87 USP30 (0.56) LMNASTSGPR119BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116615427-A Substituted macrocyclic compounds and related methods of treatment 阿尔克姆斯有限公司 2023-08-18 CN disclosed
CN-114761412-A Substituted macrocyclic compounds and related methods of treatment 阿尔克姆斯有限公司 2022-07-15 CN disclosed