SCHEMBL29802407

SCHEMBL29802407

CS(=O)(=O)c1ccc(-c2ccc3cc[nH]c3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.48
PTGS2 P35354 7/20 0.43
BPTF Q12830 1/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
HDAC6 Q9UBN7 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
GRM2 Q14416 1/20 0.39
IKBKB O14920 1/20 0.38
CHUK O15111 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739133 1.00 BRD4 (0.48) BRD4PTGS2BPTFMAOAMAOB
SCHEMBL416127 0.76 APP (0.50)
SCHEMBL31065010 0.75 RIPK1 (0.54) BRD4NPC1ALDH1A1RAB9A
SCHEMBL16417014 0.75 MAPK1 (0.54) BRD4MAOAMAOBKDM4ENPC1
SCHEMBL16416975 0.75 AXL (0.50) BRD4DYRK1BCDK5IKBKBCHUK
SCHEMBL14735035 0.74 BRD4 (0.53) BRD4DYRK1BCDK5IKBKBCHUK
SCHEMBL23110560 0.74 BRD4 (0.50) BRD4PTGS2
SCHEMBL16417052 0.74 BRD4 (0.50) BRD4MAOAMAOBALDH1A1
SCHEMBL16417000 0.74 BRD4 (0.61) BRD4KDM4ENPC1ALDH1A1RAB9A
SCHEMBL857607 0.73 RIPK1 (0.61) BRD4DYRK1BCDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4027993-A1 CYCLOOXYGENASE-2 INHIBITORS AND USES THEREOF The Broad Institute Inc. (US) 2022-07-20 EP disclosed