SCHEMBL29804259

SCHEMBL29804259

N[C@@H](Cc1c[nH]c2ccc(O)cc12)C(=O)NCCc1c[nH]c2ccc(O)cc12

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.77
SPR P35270 4/20 0.74
KDM4E B2RXH2 4/20 0.67
ALDH1A1 P00352 3/20 0.67
NPSR1 Q6W5P4 3/20 0.67
HTR2C P28335 3/20 0.67
CYP3A4 P08684 2/20 0.67
MAPT P10636 2/20 0.67
BLM P54132 2/20 0.67
LMNA P02545 2/20 0.67
HTR1A P08908 2/20 0.67
NFKB1 P19838 2/20 0.67
HTR2A P28223 2/20 0.67
HTR2B P41595 2/20 0.67
KMT2A Q03164 2/20 0.67
ADORA3 P0DMS8 1/20 0.67
ALOX15 P16050 1/20 0.67
TSHR P16473 1/20 0.67
SLC6A4 P31645 1/20 0.67
HTR7 P34969 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20168582 1.00 HDAC8 (0.77) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL20168578 1.00 HDAC8 (0.77) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL5121693 0.91 NPSR1 (0.67) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL24277478 0.91 SPR (0.74) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL6399249 0.91 SPR (0.74) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL15145410 0.90 HDAC8 (0.68) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL15145420 0.87 SPR (0.77) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL10407441 0.87 NPSR1 (0.69) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL10407439 0.87 NPSR1 (0.69) HDAC8SPRKDM4EALDH1A1NPSR1
SCHEMBL5108712 0.86 NPSR1 (0.62) HDAC8SPRKDM4EALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110177581-B Myeloperoxidase imaging agents 通用医疗公司 2023-01-03 CN disclosed
EP-4076542-A1 HIGHLY EFFICIENT MYELOPEROXIDASE ACTIVATABLE IMAGING AGENTS The General Hospital Corporation (US) 2022-10-26 EP disclosed
CN-114828900-A High efficiency myeloperoxidase activatable imaging agents 总医院公司 2022-07-29 CN disclosed