SCHEMBL2980702

SCHEMBL2980702

COc1c(Nc2ccc3[nH]ccc3c2)cccc1OCCCl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 2/20 0.45
NAE1 Q13564 1/20 0.45
JAK2 O60674 1/20 0.43
NOTUM Q6P988 2/20 0.42
EGFR P00533 3/20 0.42
ERBB2 P04626 1/20 0.42
SYK P43405 3/20 0.41
PRKCQ Q04759 2/20 0.40
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
FLT1 P17948 1/20 0.39
MAPK14 Q16539 1/20 0.37
RET P07949 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2980622 0.87 NR4A2 (0.46) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL4246552 0.86 NAE1 (0.51) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL2989022 0.85 JAK2 (0.41) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL2984052 0.85 JAK2 (0.41) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL2975051 0.84 HTR1A (0.50) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL17255750 0.84 EGFR (0.44) ULK1NAE1JAK2NOTUMEGFR
SCHEMBL2983509 0.83 HTR1A (0.51) JAK2
SCHEMBL17255760 0.83 LTA4H (0.45) JAK2NOTUMEGFRERBB2PRKCQ
SCHEMBL17255759 0.82 HTR1A (0.46) JAK2EGFRSYKPRKCQFLT1
SCHEMBL17255756 0.81 EGFR (0.42) ULK1NAE1JAK2EGFRSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781591-B2 Substituted 3-cyanopyridines as protein kinase inhibitors WYETH LLC (US) 2010-08-24 US claimed