SCHEMBL29809657

SCHEMBL29809657

O=c1[nH]ccc2cc(F)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 2/20 0.53
PARP1 P09874 2/20 0.53
GRM5 P41594 1/20 0.51
ROCK2 O75116 3/20 0.48
DAO P14920 1/20 0.46
ROCK1 Q13464 4/20 0.45
PRKACA P17612 1/20 0.45
PRKCD Q05655 1/20 0.45
PRKG1 Q13976 1/20 0.45
PKN1 Q16512 1/20 0.45
PKN2 Q16513 1/20 0.45
AAK1 Q2M2I8 1/20 0.45
CDC42BPA Q5VT25 1/20 0.45
Q6ZSR9 Q6ZSR9 1/20 0.45
BMP2K Q9NSY1 1/20 0.45
CDC42BPB Q9Y5S2 1/20 0.45
CHEK1 O14757 1/20 0.44
TYMS P04818 1/20 0.44
JAK2 O60674 4/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1551818 1.00 AHR (0.53) AHRPARP1GRM5ROCK2DAO
SCHEMBL30673402 0.84 PARP1 (0.53) AHRPARP1DAOROCK1PRKACA
SCHEMBL1536413 0.84 PARP1 (0.53) AHRPARP1DAOROCK1PRKACA
SCHEMBL5983565 0.83 JAK2 (0.41) AHRPARP1GRM5ROCK2CHEK1
SCHEMBL23416327 0.83 ROCK2 (0.45) AHRPARP1GRM5ROCK2ROCK1
SCHEMBL6922954 0.81 PRKACA (0.53) PARP1GRM5ROCK2PRKACACHEK1
SCHEMBL2052887 0.78 GRM5 (0.74) PARP1GRM5ROCK2JAK2
SCHEMBL3314460 0.78 GPR84 (0.52) PARP1GRM5ROCK2ROCK1PRKACA
SCHEMBL25009087 0.77 HTR2C (0.46) PARP1GRM5ROCK2ROCK1PRKACA
SCHEMBL6797681 0.76 PARP1 (0.53) PARP1GRM5ROCK2ROCK1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114805204-A Method for preparing 4-iodoisoquinoline-1 (2H) -ketone compound 云南师范大学 2022-07-29 CN claimed
CN-113923988-B Substituted arylmethyl ureas and heteroarylmethyl ureas, analogs thereof, and methods of using the same 爱彼特生物制药公司 2024-12-13 CN disclosed
CN-118451079-A Benzopiperidine derivative modulators, methods of preparation and uses thereof 上海翰森生物医药科技有限公司 2024-08-06 CN disclosed
CN-114805204-B Method for preparing 4-iodoisoquinoline-1 (2H) -ketone compound 云南师范大学 2023-09-15 CN disclosed
CN-114805204-A Method for preparing 4-iodoisoquinoline-1 (2H) -ketone compound 云南师范大学 2022-07-29 CN disclosed