SCHEMBL29815

SCHEMBL29815

Cn1cccc1C(=O)N1CCN(C(=O)Nc2ccc(C3NCCC3CCn3cncn3)cc2)CC1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 16/20 0.66
CYP3A4 P08684 4/20 0.44
ALDH1A1 P00352 2/20 0.43
USP2 O75604 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP1A2 P05177 2/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28504 0.81 HPGDS (0.92) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL27313 0.80 HPGDS (1.00) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL28180 0.77 HPGDS (1.00) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL28360 0.69 HPGDS (1.00) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL14119527 0.67 HPGDS (0.69) HPGDS
SCHEMBL27841 0.67 HPGDS (1.00) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL28514 0.67 HPGDS (1.00) HPGDSCYP3A4
SCHEMBL15529782 0.65 HPGDS (0.53) HPGDSCYP3A4CYP1A2TSHR
SCHEMBL28861 0.65 HPGDS (0.71) HPGDSCYP3A4ALDH1A1USP2SMN1; SMN2
SCHEMBL27787 0.64 HPGDS (1.00) HPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2407466-A1 PIPERAZINE COMPOUND CAPABLE OF INHIBITING PROSTAGLANDIN D SYNTHASE Taiho Pharmaceutical Co., Ltd. (JP) 2012-01-18 EP disclosed