SCHEMBL298159

SCHEMBL298159

CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2n[nH]c3ncc(C#N)cc23)c1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.61
CYP3A4 P08684 3/20 0.61
CYP2C19 P33261 3/20 0.61
BRAF P15056 8/20 0.56
MAP2K4 P45985 7/20 0.56
BMPR1B O00238 1/20 0.56
PLK4 O00444 1/20 0.56
PIR O00625 1/20 0.56
AURKA O14965 1/20 0.56
DCLK1 O15075 1/20 0.56
EPHB6 O15197 1/20 0.56
RIPK2 O43353 1/20 0.56
STK16 O75716 1/20 0.56
OXSR1 O95747 1/20 0.56
MAP4K4 O95819 1/20 0.56
ABL1 P00519 1/20 0.56
RAF1 P04049 1/20 0.56
LCK P06239 1/20 0.56
FYN P06241 1/20 0.56
FES P07332 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21223003 0.87 BRAF (0.58) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL29915108 0.84 CYP2C19 (0.84) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL30694407 0.84 MAP2K4 (0.75) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL21223018 0.84 MAP2K4 (0.75) CYP2C19BRAFMAP2K4RIPK2RAF1
SCHEMBL30636752 0.84 MAP2K4 (0.75) CYP2C19BRAFMAP2K4RIPK2RAF1
SCHEMBL23098899 0.84 MAP2K4 (0.75) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL297652 0.84 CYP2C19 (0.84) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL21222990 0.84 MAP2K4 (0.75) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL23098883 0.84 MAP2K4 (0.66) CYP2C9CYP3A4CYP2C19BRAFMAP2K4
SCHEMBL23089255 0.84 MAP2K4 (0.65) CYP2C9CYP3A4CYP2C19BRAFMAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed