SCHEMBL298205

SCHEMBL298205

CS(=O)(=O)c1cccc(-c2cnc3[nH]cc(C(=O)c4cc(NS(=O)(=O)C5CCCC5)ccc4F)c3c2)c1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAMKK2 Q96RR4 2/20 0.49
RIPK1 Q13546 1/20 0.47
CYP2C9 P11712 4/20 0.46
CYP2C19 P33261 3/20 0.45
PAK1 Q13153 2/20 0.44
BRAF P15056 3/20 0.43
CYP3A4 P08684 2/20 0.42
PLK4 O00444 2/20 0.42
CYP2D6 P10635 1/20 0.42
PIK3CA P42336 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298881 0.99 CAMKK2 (0.48) CAMKK2RIPK1CYP2C9CYP2C19PAK1
SCHEMBL298879 0.91 CYP2C9 (0.49) RIPK1CYP2C9CYP2C19PAK1BRAF
SCHEMBL298320 0.91 CYP2C9 (0.48) RIPK1CYP2C9CYP2C19PAK1BRAF
SCHEMBL298449 0.89 CYP2C9 (0.53) CAMKK2RIPK1CYP2C9CYP2C19BRAF
SCHEMBL10246345 0.88 CYP2C19 (0.43) CYP2C9CYP2C19PAK1BRAFCYP3A4
SCHEMBL298745 0.87 CAMKK2 (0.52) CAMKK2RIPK1CYP2C9CYP2C19PAK1
SCHEMBL10246332 0.87 PAK1 (0.41) CYP2C9CYP2C19PAK1BRAFCYP3A4
SCHEMBL10246625 0.86 BRAF (0.42) RIPK1CYP2C9CYP2C19PAK1BRAF
SCHEMBL10247915 0.86 MAP2K4 (0.43) RIPK1CYP2C9CYP2C19PAK1BRAF
SCHEMBL299098 0.83 CYP3A4 (0.51) CAMKK2RIPK1CYP2C9CYP2C19BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed