SCHEMBL298879

SCHEMBL298879

CS(=O)(=O)Nc1cccc(-c2cnc3[nH]cc(C(=O)c4cc(NS(=O)(=O)C5CCCC5)ccc4F)c3c2)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 2/20 0.49
TNIK Q9UKE5 5/20 0.47
BRAF P15056 3/20 0.45
MAP2K4 P45985 1/20 0.44
PAK1 Q13153 1/20 0.43
PIK3CA P42336 1/20 0.43
CYP2D6 P10635 1/20 0.42
CLK1 P49759 1/20 0.41
DYRK1A Q13627 1/20 0.41
DYRK2 Q92630 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
CYP3A4 P08684 1/20 0.41
RIPK1 Q13546 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298320 0.99 CYP2C9 (0.48) CYP2C9CYP2C19TNIKBRAFMAP2K4
SCHEMBL298205 0.91 CAMKK2 (0.49) CYP2C9CYP2C19BRAFPAK1PIK3CA
SCHEMBL297360 0.91 CYP2C9 (0.56) CYP2C9CYP2C19TNIKBRAFPIK3CA
SCHEMBL298881 0.91 CAMKK2 (0.48) CYP2C9CYP2C19BRAFMAP2K4PAK1
SCHEMBL10246625 0.90 BRAF (0.42) CYP2C9CYP2C19BRAFMAP2K4PAK1
SCHEMBL10247915 0.90 MAP2K4 (0.43) CYP2C9CYP2C19BRAFMAP2K4PAK1
SCHEMBL10246345 0.88 CYP2C19 (0.43) CYP2C9CYP2C19BRAFMAP2K4PAK1
SCHEMBL10246332 0.88 PAK1 (0.41) CYP2C9CYP2C19BRAFMAP2K4PAK1
SCHEMBL299603 0.85 CYP2C9 (0.53) CYP2C9CYP2C19TNIKBRAFCYP2D6
SCHEMBL415675 0.85 CYP2C9 (0.52) CYP2C9CYP2C19TNIKBRAFPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed