SCHEMBL2983863

SCHEMBL2983863

CC(Oc1cncc(Br)c1)N1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.43
CHRNA4 P43681 3/20 0.43
TACR1 P25103 1/20 0.34
SLC6A4 P31645 1/20 0.34
KCNH2 Q12809 1/20 0.34
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB3 Q05901 1/20 0.33
CHRNA6 Q15825 1/20 0.33
IDH1 O75874 1/20 0.32
MC4R P32245 1/20 0.32
PIM1 P11309 1/20 0.32
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
PIM3 Q86V86 1/20 0.32
PIM2 Q9P1W9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6634 0.73 CHRNB2 (0.43) CHRNB2CHRNA4CYP11B1CYP11B2CHRNB4
SCHEMBL19417497 0.72 CHRNB2 (0.43) CHRNB2CHRNA4TACR1SLC6A4KCNH2
SCHEMBL6832889 0.71 CHRNB2 (0.39) CHRNB2CHRNA4KCNH2
SCHEMBL2936683 0.71 CHRNB2 (0.51) CHRNB2CHRNA4
SCHEMBL15206156 0.70 CHRNB2 (0.50) CHRNB2CHRNA4CYP11B2
SCHEMBL1605130 0.70 CHRNB2 (0.41) CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL7840485 0.69 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL7842116 0.69 CHRNB2 (0.42) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL23283358 0.68 CHRNB2 (0.40) CHRNB2CHRNA4
SCHEMBL28181927 0.68 CHRNB2 (0.43) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed