SCHEMBL298411

SCHEMBL298411

CCCC(c1ccc(C(N)=O)cc1C(=O)c1c[nH]c2ncc(-c3cnn(C)c3)cc12)S(=O)(=O)O

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PAK1 Q13153 14/20 0.48
CYP2C19 P33261 2/20 0.40
ALK Q9UM73 1/20 0.40
PAK4 O96013 1/20 0.39
PDPK1 O15530 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAP3K11 Q16584 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298168 0.94 PAK1 (0.49) PAK1CYP2C19ALKPAK4PDPK1
SCHEMBL299033 0.84 BRAF (0.46) PAK1CYP2C19
SCHEMBL298248 0.80 PAK1 (0.56) PAK1CYP2C19ALKPAK4MKNK1
SCHEMBL298435 0.79 PAK1 (0.51) PAK1ALKPAK4MKNK1MKNK2
SCHEMBL297658 0.79 DYRK1A (0.43) PAK1PAK4PDPK1MKNK1MKNK2
SCHEMBL299489 0.78 PAK1 (0.49) PAK1ALKPAK4PDPK1MKNK1
SCHEMBL3704923 0.77 PAK1 (0.56) PAK1ALKPAK4PDPK1MKNK1
SCHEMBL299284 0.77 BRAF (0.45) PAK1CYP2C19
SCHEMBL298640 0.77 BRAF (0.37) PAK1CYP2C19PAK4PDPK1MAP3K11
SCHEMBL28481416 0.74 PDPK1 (0.51) PAK1ALKPDPK1MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed