SCHEMBL29849232

SCHEMBL29849232

COc1ccc(CNc2ncnc(Cl)c2C=O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.55
EGFR P00533 4/20 0.53
POLB P06746 2/20 0.53
NR2F2 P24468 1/20 0.53
LMNA P02545 2/20 0.52
ALDH1A1 P00352 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
PDE5A O76074 1/20 0.51
THRB P10828 1/20 0.49
MAPT P10636 3/20 0.48
TP53 P04637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
CDK1 P06493 3/20 0.48
CCNB2 O95067 2/20 0.48
CCNB1 P14635 2/20 0.48
CCNB3 Q8WWL7 2/20 0.48
AURKA O14965 1/20 0.47
RPS6KB1 P23443 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29060167 1.00 HTT (0.55) HTTEGFRPOLBNR2F2LMNA
SCHEMBL19305769 0.87 HTT (0.55) HTTEGFRPOLBNR2F2LMNA
SCHEMBL29059871 0.83 HTT (0.49) HTTEGFRPOLBNR2F2LMNA
SCHEMBL29849114 0.83 HTT (0.49) HTTEGFRPOLBNR2F2LMNA
SCHEMBL29956286 0.82 EGFR (0.50) HTTEGFRNR2F2LMNAALDH1A1
SCHEMBL24096410 0.81 CA1 (0.50) HTTEGFRPOLBNR2F2ALDH1A1
SCHEMBL29634669 0.80 HTT (0.58) HTTEGFRPOLBNR2F2LMNA
SCHEMBL5233252 0.80 HTT (0.58) HTTEGFRPOLBNR2F2LMNA
SCHEMBL16781105 0.79 LMNA (0.58) HTTEGFRPOLBNR2F2LMNA
SCHEMBL20061415 0.79 HTT (0.54) HTTEGFRPOLBNR2F2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116669738-A Pyrimidopyridone derivative as SOS1 inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2023-08-29 CN disclosed
WO-2022170802-A1 PYRIMIDO-PYRIDONE DERIVATIVE AS SOS1 INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF 苏州阿尔脉生物科技有限公司 2022-08-18 WO disclosed