SCHEMBL29860906

SCHEMBL29860906

CC(=O)c1ccc(NC(=O)C2C(C)(C)C2(C)C)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCK P35557 2/20 0.43
WNT1 P04628 2/20 0.43
GSK3B P49841 2/20 0.43
DYRK1A Q13627 2/20 0.43
HCAR3 P49019 5/20 0.42
TSHR P16473 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PTK2 Q05397 1/20 0.41
NNMT P40261 1/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 2/20 0.40
MAPT P10636 1/20 0.40
TP53 P04637 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
DEGS1 O15121 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29854816 0.82 GCK (0.40) GCKWNT1GSK3BDYRK1AHCAR3
SCHEMBL28810935 0.82 GCK (0.40) GCKWNT1GSK3BDYRK1AHCAR3
SCHEMBL24932386 0.81 DEGS1 (0.53) DEGS1
SCHEMBL24932388 0.81 RAB9A (0.64) NPSR1GAARAB9AMAPTTP53
SCHEMBL7093993 0.80 PTK2 (0.62) HCAR3TSHRPTK2NNMTCYP1A2
SCHEMBL24932390 0.79 PTK2 (0.63) TSHRNPSR1PTK2RAB9AMAPT
SCHEMBL24932387 0.79 WNT1 (0.43) WNT1GSK3BDYRK1ATSHRNPSR1
SCHEMBL24932289 0.79 KDM4E (0.47) WNT1GSK3BDYRK1ARAB9ASMN1; SMN2
SCHEMBL29854902 0.78 MAPT (0.43) GCKWNT1GSK3BDYRK1ACYP1A2
SCHEMBL28811296 0.78 MAPT (0.43) GCKWNT1GSK3BDYRK1ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901280-A MrgprX2 antagonists and uses thereof 德米拉公司 2022-08-12 CN disclosed