SCHEMBL29863239

SCHEMBL29863239

COCC(=O)N1Cc2ccccc2N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.40
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 2/20 0.38
MAPK1 P28482 3/20 0.37
CYP2D6 P10635 5/20 0.36
TAAR1 Q96RJ0 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 5/20 0.36
USP2 O75604 3/20 0.36
HSD17B3 P37058 1/20 0.35
TP53 P04637 1/20 0.35
HIF1A Q16665 1/20 0.35
NOTUM Q6P988 1/20 0.35
CYP2C19 P33261 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29863425 0.81 BRD4 (0.39) NAMPTBRD4CREBBPMAPK1SMN1; SMN2
SCHEMBL4880946 0.77 BRD4 (0.45) NAMPTBRD4CREBBPALDH1A1MAPK1
SCHEMBL5822563 0.75 BRD4 (0.42) BRD4CREBBPALDH1A1MAPK1SMN1; SMN2
SCHEMBL30125059 0.75 BRD4 (0.42) BRD4CREBBPALDH1A1MAPK1SMN1; SMN2
SCHEMBL29491264 0.67 BRD4 (0.41) NAMPTBRD4CREBBPALDH1A1CYP1A2
SCHEMBL25422279 0.65 BRD4 (0.39) BRD4CREBBPALDH1A1CYP1A2MAPK1
SCHEMBL3458566 0.65 ALDH1A1 (0.41) NAMPTALDH1A1CYP1A2CYP2D6SMN1; SMN2
Indoline SCHEMBL8922922 0.64 MAPK1 (0.40) BRD4ALDH1A1CYP1A2MAPK1SMN1; SMN2
SCHEMBL13239096 0.63 BRD4 (0.52) BRD4CREBBPALDH1A1MAPK1SMN1; SMN2
SCHEMBL27881241 0.63 BRD4 (0.43) BRD4CREBBPALDH1A1CYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901279-A Inhibitors of cGAS for the treatment of autoinflammatory diseases and cancer metastasis 洛克菲勒大学 2022-08-12 CN disclosed