SCHEMBL29869232

SCHEMBL29869232

C/C=C\C=C\C=C\c1cc(N2c3ccccc3-c3ccc(-c4ccccc4C(=O)OC)c4cccc2c34)nc(-c2ccccc2)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.33
TSHR P16473 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
GRM5 P41594 1/20 0.31
TOP2A P11388 1/20 0.31
ABCC1 P33527 1/20 0.30
ABCG2 Q9UNQ0 1/20 0.30
ROCK2 O75116 1/20 0.30
CSF1R P07333 1/20 0.30
KDR P35968 1/20 0.30
FLT3 P36888 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
ROCK1 Q13464 1/20 0.30
SLK Q9H2G2 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30
USP30 Q70CQ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21073902 1.00 PDE5A (0.33) PDE5ATSHRSLC6A2SLC6A4SLC6A3
SCHEMBL30343471 1.00 PDE5A (0.33) PDE5ATSHRSLC6A2SLC6A4SLC6A3
SCHEMBL19980354 0.85 PLA2G2A (0.39) PDE5ATSHRSLC6A2SLC6A4SLC6A3
SCHEMBL21073901 0.81 GRM5 (0.33) PDE5ATSHRSLC6A2SLC6A4SLC6A3
SCHEMBL19980357 0.76 GRM5 (0.42) TSHRSLC6A2SLC6A4SLC6A3GRM5
SCHEMBL19980356 0.72 TSHR (0.41) TSHRSLC6A2SLC6A4SLC6A3TOP2A
SCHEMBL13324417 0.65 SLC6A3 (0.50) TSHRSLC6A2SLC6A4SLC6A3ROCK2
SCHEMBL19974401 0.64 HPGD (0.42) TSHR
SCHEMBL21942516 0.63 SLC6A3 (0.43) TSHRSLC6A2SLC6A4SLC6A3GRM5
SCHEMBL24891060 0.62 MYC (0.49) TSHRSLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11447464-B2 Compounds with spirobifluorene-structures MERCK PATENT GMBH (DE) 2022-09-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11447464-B2 Compounds with spirobifluorene-structures SLCO1B3, SLCO4C1, SLCO1B1 PDE5A 3310/4885TSHR 3504/4885SLC6A2 29/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.