SCHEMBL2987634

SCHEMBL2987634

CC(C)N(C)[C@@H]1CC[C@H](NC(=O)OCc2ccccc2)[C@@H](CS(=O)(=O)c2ccc(Br)cc2)C1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 18/20 0.55
CYP2D6 P10635 1/20 0.51
KCNH2 Q12809 2/20 0.45
CPB1 P15086 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2987631 1.00 CCR2 (0.55) CCR2CYP2D6KCNH2CPB1
SCHEMBL3425020 0.92 CCR2 (0.54) CCR2CYP2D6KCNH2
SCHEMBL3425012 0.92 CCR2 (0.54) CCR2CYP2D6KCNH2
SCHEMBL3427499 0.90 CCR2 (0.50) CCR2CYP2D6KCNH2CPB1
SCHEMBL3427501 0.90 CCR2 (0.50) CCR2CYP2D6KCNH2CPB1
SCHEMBL3427504 0.90 CCR2 (0.50) CCR2CYP2D6KCNH2CPB1
SCHEMBL2989537 0.85 CCR2 (0.50) CCR2KCNH2CPB1
SCHEMBL2992417 0.85 CCR2 (0.50) CCR2KCNH2CPB1
SCHEMBL2992421 0.85 CCR2 (0.50) CCR2KCNH2CPB1
SCHEMBL2989535 0.85 CCR2 (0.50) CCR2KCNH2CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776884-B2 Cyclic derivatives as modulators of chemokine receptors activity BRISTOL-MYERS SQUIBB COMPANY (US) 2010-08-17 US disclosed
US-7087604-B2 Cyclic derivatives as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2006-08-08 US disclosed