SCHEMBL29878486

SCHEMBL29878486

N#Cc1ccc2c(c1)CC(Nc1ncc(Br)cn1)C2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 1/20 0.41
PNMT P11086 6/20 0.37
GRIA2 P42262 1/20 0.36
ENPP2 Q13822 1/20 0.36
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
DRD2 P14416 2/20 0.34
DRD3 P35462 2/20 0.34
IRAK4 Q9NWZ3 2/20 0.34
CSNK2A1 P68400 1/20 0.34
MCHR1 Q99705 2/20 0.34
CCNT1 O60563 1/20 0.33
CCNK O75909 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
CDK12 Q9NYV4 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23519606 1.00 IDH1 (0.41) IDH1PNMTGRIA2ENPP2HDAC8
SCHEMBL23501018 0.82 ENPP2 (0.42) IDH1ENPP2HDAC8HDAC6CCNK
SCHEMBL29878779 0.79 NAMPT (0.45) IDH1GRIA2HDAC8HDAC6CCNK
SCHEMBL23500959 0.79 NAMPT (0.45) IDH1GRIA2HDAC8HDAC6CCNK
SCHEMBL24112177 0.79 MAPK1 (0.39) IDH1GRIA2ENPP2HDAC8HDAC6
SCHEMBL24112178 0.79 MAPK1 (0.39) IDH1GRIA2ENPP2HDAC8HDAC6
SCHEMBL22057917 0.78 ENPP2 (0.48) ENPP2
SCHEMBL29771574 0.78 ENPP2 (0.48) ENPP2
SCHEMBL22057213 0.77 KDM4E (0.46) ENPP2CSNK2A1
SCHEMBL30807501 0.77 KDM4E (0.46) ENPP2CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114901658-A Nitrogen-containing heterocyclic ring autotaxin inhibitor, and composition and application thereof 四川海思科制药有限公司 2022-08-12 CN disclosed