SCHEMBL29891877

SCHEMBL29891877

N#Cc1ccc2[nH]c(=O)c(C#N)cc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.51
IMPDH1 P20839 1/20 0.51
CYP19A1 P11511 2/20 0.51
CHEK1 O14757 2/20 0.45
IDH1 O75874 5/20 0.45
FASN P49327 1/20 0.43
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
MAPK10 P53779 1/20 0.41
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
KDM4E B2RXH2 2/20 0.40
GALR3 O60755 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19751545 0.81 DAO (0.58) IDH1KDM4EGALR3ALDH1A1GAA
SCHEMBL7264461 0.81 IDH1 (0.51) CYP19A1CHEK1IDH1KDM4EGALR3
SCHEMBL10691248 0.81 DAO (0.58) IDH1
SCHEMBL8139952 0.81 FLT3 (0.49) CHEK1IDH1CA2GAANPSR1
SCHEMBL22185219 0.81 BRD4 (0.54) IMPDH2IMPDH1CYP19A1CHEK1IDH1
SCHEMBL10690995 0.79 KDM4E (0.43) IDH1KDM4EGALR3ALDH1A1GAA
SCHEMBL1903750 0.79 BRD4 (0.55) CHEK1IDH1CA1CA2KDM4E
SCHEMBL29890500 0.79 BRD4 (0.55) CHEK1IDH1CA1CA2KDM4E
SCHEMBL7499153 0.78 IDH1 (0.58) IDH1CA2KDM4EALDH1A1GAA
SCHEMBL7501391 0.78 IDH1 (0.55) IDH1KDM4EGALR3ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115003665-A Substituted aminoquinolones as immunoactive DGK alpha inhibitors 拜耳公司 2022-09-02 CN disclosed