SCHEMBL29893178

SCHEMBL29893178

O=[N+]([O-])c1cccc(N(Cc2ccccc2)Cc2ccccc2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60
CYP2C19 P33261 1/20 0.60
ALDH1A1 P00352 5/20 0.59
PKM P14618 2/20 0.59
KDM4E B2RXH2 2/20 0.59
HTT P42858 1/20 0.59
LMNA P02545 4/20 0.57
CRHBP P24387 3/20 0.53
CRHR2 Q13324 3/20 0.53
TSHR P16473 2/20 0.51
PTPN1 P18031 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
NR3C1 P04150 1/20 0.48
FAAH O00519 1/20 0.47
MGLL Q99685 1/20 0.47
NPC1 O15118 1/20 0.47
CASP3 P42574 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11788916 1.00 CYP1A2 (0.60) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL18138825 0.91 ALDH1A1 (0.57) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL28067958 0.88 CYP1A2 (0.57) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL11789106 0.84 CRHBP (0.70) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL18300788 0.84 ALDH1A1 (0.54) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL18300787 0.84 ALDH1A1 (0.54) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL18138735 0.83 ALDH1A1 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL18138736 0.83 ALDH1A1 (0.53) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL8537467 0.81 CRHBP (0.61) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL627381 0.81 CRHBP (0.71) CYP1A2CYP2D6CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313308-A1 TEAD INHIBITORS AND USES THEREOF Cedilla Therapeutics, Inc. (US) 2024-02-07 EP disclosed
WO-2022204452-A1 TEAD INHIBITORS AND USES THEREOF CEDILLA THERAPEUTICS, INC. (US) 2022-09-29 WO disclosed