SCHEMBL29897243

SCHEMBL29897243

c1cncc(-c2cc(C3CC3)on2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.55
CYP2A6 P11509 3/20 0.55
NPC1 O15118 3/20 0.55
CYP2E1 P05181 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2B6 P20813 1/20 0.55
CYP2C19 P33261 1/20 0.55
PPARA Q07869 1/20 0.48
CHRNB2 P17787 1/20 0.46
CHRNA5 P30532 1/20 0.46
CHRNA4 P43681 1/20 0.46
KDM4E B2RXH2 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HPGDS O60760 1/20 0.44
TP53 P04637 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
USP30 Q70CQ3 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11835580 1.00 RAB9A (0.55) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL4919930 0.88 CYP2A6 (0.50) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL3853565 0.82 CYP2C9 (0.47) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL11783495 0.81 RAB9A (0.54) RAB9ANPC1CYP2C9CYP2C19USP30
SCHEMBL4036212 0.81 CHRNB2 (0.54) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL11836452 0.80 NPC1 (0.45) RAB9ANPC1CYP1A2
SCHEMBL14466141 0.78 CYP2C9 (0.46) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL14466245 0.78 CYP2C9 (0.46) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL11841512 0.76 SCD (0.50) RAB9ACYP2A6NPC1CYP2E1CYP2C9
SCHEMBL4318440 0.76 CYP3A4 (0.62) RAB9ACYP2A6NPC1CYP2E1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111615514-B Substituted pyrazolo [4,3-C ] pyridine compounds as RET kinase inhibitors 奥瑞生物药品公司 2022-10-11 CN disclosed