SCHEMBL29901586

SCHEMBL29901586

C#CCN1C(=O)C(C)(C)Oc2cc(F)c(N)cc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
RECQL P46063 1/20 0.39
NR3C2 P08235 1/20 0.36
KMT2A Q03164 3/20 0.35
POLB P06746 2/20 0.35
PGR P06401 1/20 0.35
MEN1 O00255 1/20 0.34
REN P00797 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16541627 0.89 PGR (0.34) ALDH1A1PGR
SCHEMBL30704859 0.87 PGR (0.32) ALDH1A1PGR
SCHEMBL900663 0.87 PGR (0.32) ALDH1A1PGR
SCHEMBL28062084 0.85 PGR (0.31) ALDH1A1PGR
SCHEMBL20692934 0.84 NR3C2 (0.34) ALDH1A1NR3C2PGRREN
SCHEMBL25362198 0.82 ALDH1A1 (0.37) ALDH1A1MAPTRECQLNR3C2KMT2A
SCHEMBL30799184 0.82 NR3C2 (0.36) ALDH1A1NR3C2REN
SCHEMBL20693048 0.82 NR3C2 (0.36) ALDH1A1NR3C2REN
SCHEMBL30193857 0.82 ALDH1A1 (0.37) ALDH1A1MAPTRECQLNR3C2KMT2A
SCHEMBL26001531 0.79 ALDH1A1 (0.37) ALDH1A1MAPTRECQLNR3C2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113200985-B Pteridinone compound and preparation method and application thereof 南开大学 2022-09-09 CN disclosed