SCHEMBL2990200

SCHEMBL2990200

O=C(O)Cc1ccc(Oc2ccc(C(=O)NC(Cl)Cc3ccc(Cl)cc3)cc2)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 3/20 0.44
FFAR1 O14842 2/20 0.42
PTGDR2 Q9Y5Y4 4/20 0.42
PPARD Q03181 2/20 0.42
PPARA Q07869 2/20 0.42
PPARG P37231 1/20 0.42
PTGDR Q13258 2/20 0.41
CA2 P00918 1/20 0.41
SRD5A2 P31213 1/20 0.40
PNLIP P16233 1/20 0.40
PTGER4 P35408 1/20 0.40
THRA P10827 2/20 0.39
THRB P10828 2/20 0.39
PTPN1 P18031 1/20 0.39
MMP1 P03956 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2982722 0.85 PTGDR2 (0.51) FFAR1PTGDR2PPARDPPARAPPARG
SCHEMBL2991855 0.82 GAA (0.54) PTGDR2PPARDPPARAPPARGTHRA
SCHEMBL2990197 0.77 TRPV1 (0.56) NR3C1FFAR1PTGDR2PTGDR
SCHEMBL13742693 0.74 KDM4E (0.67) PTGDR2PNLIP
SCHEMBL13742653 0.73 PNLIP (0.67) FFAR1PTGDR2PTGDRPNLIP
SCHEMBL1569817 0.72 RAB9A (0.56) PPARGCA2
SCHEMBL2986773 0.72 PTGDR2 (0.40) PTGDR2PPARAPPARGPTGDRSRD5A2
SCHEMBL2982709 0.72 PTGDR2 (0.60) FFAR1PTGDR2PPARDPPARAPPARG
SCHEMBL13742473 0.71 TRPV1 (0.53) PTGDR2
SCHEMBL4078169 0.71 MCHR1 (0.55) PTGDR2PPARDPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8492437-B2 4-substituted phenoxyphenylacetic acid derivatives ARRAY BIOPHARMA INC. (US) 2013-07-23 US claimed
US-20120202854-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2012-08-09 US claimed
US-8492437-B2 4-substituted phenoxyphenylacetic acid derivatives ARRAY BIOPHARMA INC. (US) 2013-07-23 US disclosed
EP-2057115-B9 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC (US) 2012-12-26 EP disclosed
EP-2057115-B1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC (US) 2012-10-03 EP disclosed
US-20120202854-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2012-08-09 US disclosed
US-8183289-B2 4-substituted phenoxyphenylacetic acid derivatives ARRAY BIOPHARMA INC. (US) 2012-05-22 US disclosed
US-20100173955-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA INC. (US) 2010-07-08 US disclosed
EP-2057115-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES Array Biopharma, Inc. (US) 2009-05-13 EP disclosed
WO-2008024746-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES ARRAY BIOPHARMA, INC. (US) 2008-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100173955-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES CD22, HRH2, CD74 NR3C1 262/4885FFAR1 87/4885PTGDR2 12/4885
US-20120202854-A1 4-SUBSTITUTED PHENOXYPHENYLACETIC ACID DERIVATIVES CD22, HRH2, CD74 NR3C1 262/4885FFAR1 87/4885PTGDR2 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.