SCHEMBL29902509

SCHEMBL29902509

Cn1cc(-c2ccc(F)cc2)c(=O)c(C(N)=O)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1D P48730 5/20 0.48
CSNK1E P49674 4/20 0.48
MAPK14 Q16539 2/20 0.48
MAPK13 O15264 1/20 0.48
MAPK12 P53778 1/20 0.48
MAPK11 Q15759 1/20 0.48
GRM2 Q14416 5/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
MAP4K4 O95819 2/20 0.40
MAPK9 P45984 2/20 0.40
CSNK1A1 P48729 2/20 0.40
EGFR P00533 1/20 0.40
FRK P42685 1/20 0.40
KCNH2 Q12809 2/20 0.39
NR1I2 O75469 1/20 0.39
NUAK1 O60285 1/20 0.39
ROCK2 O75116 1/20 0.39
LCK P06239 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23160878 0.88 CSNK1D (0.48) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL29902500 0.82 ADORA2A (0.42) CSNK1DCSNK1EGRM2KDM4EALDH1A1
SCHEMBL30499536 0.81 LMNA (0.51) MAPK14KDM4EALDH1A1HPGDADORA2A
SCHEMBL1257163 0.80 CSNK1D (0.51) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL30136520 0.79 MET (0.41) CSNK1DGRM2KDM4EALDH1A1HPGD
SCHEMBL29902513 0.78 IRAK4 (0.47) CSNK1DCSNK1EGRM2KDM4EGSK3B
SCHEMBL22309898 0.77 SLC6A4 (0.50) CSNK1DCSNK1EMAPK14MAPK13MAPK12
SCHEMBL14335004 0.75 IRAK4 (0.51) GRM2KDM4EALDH1A1HPGDADORA2A
SCHEMBL15328107 0.75 MET (0.50) GRM2METAXLPTGS1ABCB1
SCHEMBL9585904 0.73 LMNA (0.54) CSNK1DCSNK1EMAPK14MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112625027-B Heterocyclic derivatives and use thereof 药捷安康(南京)科技股份有限公司 2022-09-09 CN disclosed