SCHEMBL29907703

SCHEMBL29907703

N#Cc1cccc(N2CCCC2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 3/20 0.46
CNR1 P21554 1/20 0.44
PIM1 P11309 3/20 0.42
CTSK P43235 1/20 0.41
ALDH1A1 P00352 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 2/20 0.41
PDE10A Q9Y233 1/20 0.41
PARP1 P09874 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
LCAT P04180 1/20 0.40
NPC1 O15118 1/20 0.40
GALR3 O60755 1/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21730194 1.00 CTSS (0.46) CTSSCNR1PIM1CTSKALDH1A1
SCHEMBL2949577 0.98 CTSS (0.45) CTSSCNR1PIM1CTSKALDH1A1
SCHEMBL21730383 0.96 CTSS (0.46) CTSSCNR1PIM1CTSKALDH1A1
SCHEMBL23166854 0.89 ALDH1A1 (0.49) CTSSCNR1CTSKALDH1A1L3MBTL1
SCHEMBL15347238 0.86 PIM1 (0.53) PIM1ALDH1A1KDM4ECASP1MAPK1
SCHEMBL30077085 0.86 PIM1 (0.53) PIM1ALDH1A1KDM4ECASP1MAPK1
SCHEMBL27920871 0.86 CTSS (0.44) CTSSPIM1CTSKALDH1A1L3MBTL1
SCHEMBL21268766 0.84 ALDH1A1 (0.58) CTSSPIM1ALDH1A1KDM4EMAPK1
SCHEMBL30893584 0.84 ALDH1A1 (0.58) CTSSPIM1ALDH1A1KDM4EMAPK1
SCHEMBL2814727 0.84 LRRK2 (0.52) CTSSALDH1A1L3MBTL1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115181092-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2024-05-03 CN disclosed
CN-115181092-A Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-10-14 CN disclosed
CN-112279837-B Pyrazine compounds and uses thereof 迪哲(江苏)医药股份有限公司 2022-08-09 CN disclosed