SCHEMBL29908276

SCHEMBL29908276

O=C(Nc1ncc(Br)s1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.64
DEGS1 O15121 1/20 0.51
PTGS1 P23219 2/20 0.50
KCNQ3 O43525 1/20 0.50
KCNQ2 O43526 1/20 0.50
KCNE1 P15382 1/20 0.50
KCNQ1 P51787 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
SCD O00767 2/20 0.47
HDAC1 Q13547 1/20 0.47
NPC1 O15118 2/20 0.47
LMNA P02545 1/20 0.47
PKM P14618 1/20 0.47
RAB9A P51151 1/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47
CDK5 Q00535 1/20 0.47
MAPT P10636 1/20 0.47
XBP1 P17861 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836669 0.82 KDR (0.68) SMN1; SMN2SCDHDAC1NPC1LMNA
SCHEMBL28573896 0.79 STAT3 (1.00) STAT3SMN1; SMN2NPC1LMNAPKM
SCHEMBL27569509 0.78 HDAC1 (0.46) STAT3SMN1; SMN2SCDHDAC1NPC1
SCHEMBL5835755 0.78 CA2 (0.60) SMN1; SMN2HDAC1NPC1LMNAPKM
SCHEMBL4601021 0.76 KDR (0.46) PKMCCNE1CDK2KDR
SCHEMBL4717243 0.76 CA12 (0.49) KDR
SCHEMBL2650712 0.75 SMN1; SMN2 (0.54) SMN1; SMN2NPC1LMNAPKMRAB9A
SCHEMBL13055703 0.74 STAT3 (0.54) STAT3DEGS1SMN1; SMN2SCDNPC1
Ammonia Solution, Strong SCHEMBL27867504 0.74 SMN1; SMN2 (0.52) SMN1; SMN2NPC1LMNAPKMRAB9A
SCHEMBL25422503 0.73 RAB9A (0.55) SMN1; SMN2HDAC1NPC1LMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116456980-A Application of thiazole compounds in preparation of medicines for treating and preventing cancers 北京大学 2023-07-18 CN disclosed
WO-2022206084-A1 USE OF THIAZOLE COMPOUND IN PREPARATION OF DRUG FOR TREATING AND PREVENTING CANCER 北京大学 2022-10-06 WO disclosed