SCHEMBL29908284

SCHEMBL29908284

Cc1ccc(C(=O)Nc2ncc([N+](=O)[O-])s2)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 9/20 1.00
NPC1 O15118 11/20 0.68
RAB9A P51151 11/20 0.68
MEN1 O00255 8/20 0.68
KMT2A Q03164 8/20 0.68
PKM P14618 6/20 0.68
POLB P06746 3/20 0.59
ALDH1A1 P00352 4/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
LMNA P02545 2/20 0.58
MAPT P10636 4/20 0.56
NPSR1 Q6W5P4 2/20 0.56
MLNR O43193 1/20 0.56
NR1I2 O75469 1/20 0.56
ABCB11 O95342 1/20 0.56
TP53 P04637 1/20 0.56
ADRB2 P07550 1/20 0.56
CHRM2 P08172 1/20 0.56
ADRB1 P08588 1/20 0.56
CYP3A4 P08684 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795075 1.00 STAT3 (1.00) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL5797958 0.91 STAT3 (1.00) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL29908285 0.91 STAT3 (1.00) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL25063001 0.89 STAT3 (0.80) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL28574896 0.88 STAT3 (0.78) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL25063050 0.87 STAT3 (0.80) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL5795728 0.83 NPC1 (0.75) STAT3NPC1RAB9AMEN1KMT2A
Tizoxanide SCHEMBL375440 0.83 STAT3 (1.00) STAT3NPC1RAB9AMEN1KMT2A
Tizoxanide SCHEMBL29367981 0.83 STAT3 (1.00) STAT3NPC1RAB9AMEN1KMT2A
SCHEMBL22680776 0.81 NPC1 (1.00) STAT3NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116456980-A Application of thiazole compounds in preparation of medicines for treating and preventing cancers 北京大学 2023-07-18 CN disclosed
WO-2022206084-A1 USE OF THIAZOLE COMPOUND IN PREPARATION OF DRUG FOR TREATING AND PREVENTING CANCER 北京大学 2022-10-06 WO disclosed