SCHEMBL29908996

SCHEMBL29908996

CC(C)(C)OC(=O)N1CCC(Nc2n[nH]c3cc(Br)ccc23)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.62
ALDH1A1 P00352 2/20 0.51
NPC1 O15118 1/20 0.50
MAPT P10636 1/20 0.50
MAPK1 P28482 1/20 0.50
HTT P42858 1/20 0.50
RAB9A P51151 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NSD2 O96028 1/20 0.49
DYRK1A Q13627 3/20 0.48
IDO1 P14902 1/20 0.48
TDO2 P48775 1/20 0.48
DNMT3A Q9Y6K1 1/20 0.47
USP30 Q70CQ3 1/20 0.46
GPR119 Q8TDV5 3/20 0.45
GSK3B P49841 1/20 0.45
FPR3 P25089 1/20 0.44
FPR2 P25090 1/20 0.44
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26967728 1.00 CNR1 (0.62) CNR1ALDH1A1NPC1MAPTMAPK1
SCHEMBL29908994 1.00 CNR1 (0.62) CNR1ALDH1A1NPC1MAPTMAPK1
SCHEMBL28581769 0.84 L3MBTL1 (0.52) CNR1ALDH1A1NPC1RAB9AL3MBTL1
SCHEMBL26967715 0.84 DYRK1A (0.52) CNR1DYRK1AIDO1GSK3B
SCHEMBL31632893 0.82 ALDH1A1 (0.59) CNR1ALDH1A1NPC1MAPTMAPK1
SCHEMBL3523230 0.80 KIT (0.47) CNR1ALDH1A1MAPTDYRK1AIDO1
SCHEMBL3299990 0.80 DDB1 (0.54) CNR1ALDH1A1NPC1MAPTMAPK1
SCHEMBL2144340 0.79 IDO1 (0.45) CNR1HTTIDO1TDO2USP30
SCHEMBL31029626 0.79 IRAK4 (0.65) ALDH1A1NSD2GPR119IRAK4BTK
SCHEMBL30902132 0.79 IRAK4 (0.65) ALDH1A1NSD2GPR119IRAK4BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4294811-A2 SMALL MOLECULES THAT BIND TO TDP-43 FOR THE TREATMENT OF ALS AND RELATED DISORDERS Biohaven Therapeutics Ltd. (US) 2023-12-27 EP disclosed
WO-2022178338-A2 SMALL MOLECULES THAT BIND TO TDP-43 FOR THE TREATMENT OF ALS AND RELATED DISORDERS BIOHAVEN THERAPEUTICS LTD. (US) 2022-08-25 WO disclosed