SCHEMBL29912754

SCHEMBL29912754

COc1cccc(OCC(=O)N2CCC(Oc3ccccc3)CC2)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.66
EPHX2 P34913 1/20 0.58
KMT2A Q03164 2/20 0.55
MEN1 O00255 1/20 0.55
MAPK1 P28482 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TP53 P04637 3/20 0.54
NPC1 O15118 1/20 0.54
MAPT P10636 1/20 0.54
RAB9A P51151 1/20 0.54
ALDH1A1 P00352 5/20 0.53
LMNA P02545 2/20 0.53
RECQL P46063 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
USP2 O75604 1/20 0.52
KDM4E B2RXH2 3/20 0.51
TDP1 Q9NUW8 2/20 0.51
POLB P06746 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27158734 1.00 GAA (0.66) GAAEPHX2KMT2AMEN1MAPK1
SCHEMBL10313329 0.83 KMT2A (0.67) KMT2AMEN1MAPTPOLB
SCHEMBL791567 0.81 GAA (0.78) GAAKMT2AMEN1NPC1MAPT
SCHEMBL6445936 0.81 MEN1 (0.64) EPHX2KMT2AMEN1MAPK1SMN1; SMN2
SCHEMBL19702752 0.80 GAA (0.53) GAAEPHX2KMT2AMEN1MAPK1
SCHEMBL19702681 0.80 GAA (0.53) GAAEPHX2KMT2AMEN1MAPK1
SCHEMBL5059902 0.79 ALDH1A1 (0.78) GAAKMT2AMEN1MAPK1SMN1; SMN2
SCHEMBL2093978 0.78 EPHX2 (0.60) EPHX2KMT2AMAPK1NPC1MAPT
SCHEMBL2093973 0.77 EPHX2 (0.58) GAAEPHX2KMT2AMEN1MAPK1
SCHEMBL19852049 0.77 HRH3 (0.65) KMT2AMAPK1SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
CN-117642404-A Small molecule modulators of glucocerebrosidase activity and uses thereof 凡况生化公司 2024-03-01 CN disclosed
WO-2022232383-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2022-11-03 WO disclosed