SCHEMBL29912937

SCHEMBL29912937

Nc1nc(Cl)cnc1C#Cc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.40
GRM5 P41594 10/20 0.37
KCNH2 Q12809 1/20 0.37
ADK P55263 7/20 0.37
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29913169 0.84 ADK (0.48) RETGRM5ADK
SCHEMBL24367881 0.73 CDK2 (0.33)
SCHEMBL20977360 0.73 ALDH1A1 (0.33) GRM5
SCHEMBL18050635 0.72 CDK2 (0.35)
SCHEMBL2966822 0.70 ALDH1A1 (0.32)
SCHEMBL5777500 0.70 RET (0.39) RETGRM5KCNH2ADK
SCHEMBL30588906 0.69 MAPKAPK2 (0.35)
SCHEMBL24323977 0.69 TLR7 (0.38)
SCHEMBL13516914 0.69 GRM5 (0.43) GRM5
SCHEMBL4424103 0.69 CSNK1A1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4329881-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF Vanqua Bio, Inc. (US) 2024-03-06 EP disclosed
CN-117642404-A Small molecule modulators of glucocerebrosidase activity and uses thereof 凡况生化公司 2024-03-01 CN disclosed
WO-2022232383-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2022-11-03 WO disclosed