SCHEMBL29914764

SCHEMBL29914764

COc1cnc(-c2cccc(O)c2)cn1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 5/20 0.71
HSD17B2 P37059 5/20 0.71
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
FYN P06241 6/20 0.46
METAP2 P50579 1/20 0.45
KDM1A O60341 1/20 0.43
PIK3CA P42336 2/20 0.43
PIK3CB P42338 2/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CG P48736 2/20 0.43
RAF1 P04049 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
BRAF P15056 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21228179 1.00 HSD17B1 (0.71) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL1180306 0.84 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2C9FYN
SCHEMBL23601693 0.82 KDR (0.48) HSD17B1HSD17B2METAP2KDM1A
SCHEMBL16675784 0.80 FYN (0.49) HSD17B1HSD17B2FYN
SCHEMBL29462100 0.80 FYN (0.49) HSD17B1HSD17B2FYN
SCHEMBL24721117 0.79 IDO1 (0.48) HSD17B1HSD17B2KDM1AHDAC6
SCHEMBL5673332 0.79 HSD17B1 (0.97) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9
SCHEMBL24721383 0.78 HSD17B1 (0.41) HSD17B1HSD17B2
SCHEMBL30186373 0.78 HSD17B1 (0.79) HSD17B1HSD17B2CYP3A4CYP2C9FYN
SCHEMBL29431722 0.77 HSD17B1 (0.55) HSD17B1HSD17B2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094300-B Benzo-heteroaryl derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-09-16 CN disclosed