SCHEMBL29914770

SCHEMBL29914770

COc1cccc(C2=CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK4 Q16654 1/20 0.55
NAMPT P43490 2/20 0.54
GRM1 Q13255 9/20 0.53
GRM5 P41594 8/20 0.53
MMP2 P08253 2/20 0.49
ADAM10 O14672 1/20 0.49
MMP9 P14780 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
QDPR P09417 1/20 0.46
MMP3 P08254 1/20 0.46
HTR6 P50406 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TNK2 Q07912 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848748 1.00 PDK4 (0.55) PDK4NAMPTGRM1GRM5MMP2
SCHEMBL2954198 0.90 NAMPT (0.54) PDK4NAMPTGRM1GRM5TDP1
SCHEMBL21767871 0.88 PDK4 (0.47) PDK4NAMPTGRM1GRM5MMP2
SCHEMBL29941117 0.88 PDK4 (0.47) PDK4NAMPTGRM1GRM5MMP2
SCHEMBL13993114 0.88 PDK4 (0.53) PDK4NAMPTGRM1GRM5MMP2
SCHEMBL7831576 0.87 PDK4 (0.58) PDK4NAMPTGRM1GRM5HTR6
SCHEMBL8193684 0.87 NAMPT (0.59) PDK4NAMPTGRM1GRM5QDPR
SCHEMBL4872355 0.86 PDK4 (0.51) PDK4NAMPTGRM1GRM5HTR6
SCHEMBL29914645 0.86 PDK4 (0.57) PDK4NAMPTGRM1GRM5QDPR
SCHEMBL1364792 0.86 PDK4 (0.57) PDK4NAMPTGRM1GRM5QDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111094300-B Benzo-heteroaryl derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-09-16 CN disclosed