SCHEMBL29916533

SCHEMBL29916533

Cc1cc(C)c(Oc2nc(Cc3ccccc3)ccc2C(=O)NS(=O)(=O)c2cccc(N)n2)c(C)c1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.36
BRD4 O60885 6/20 0.35
EGFR P00533 1/20 0.34
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA2B P08514 1/20 0.33
FLT1 P17948 2/20 0.33
FLT4 P35916 2/20 0.33
KDR P35968 2/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP13 P45452 1/20 0.32
SCN9A Q15858 2/20 0.32
ADORA2A P29274 1/20 0.31
MEN1 O00255 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17649314 1.00 KLKB1 (0.36) KLKB1BRD4EGFRITGB3ITGAV
SCHEMBL17647992 0.92 ITGB3 (0.39) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL29916260 0.92 ITGB3 (0.39) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL17648601 0.89 FLT1 (0.35) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL29916998 0.89 FLT1 (0.35) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL17646540 0.85 SCN9A (0.36) KLKB1THRATHRBSCN9A
SCHEMBL29918033 0.85 SCN9A (0.36) KLKB1THRATHRBSCN9A
SCHEMBL17647642 0.85 ITGB3 (0.37) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL29916262 0.85 ITGB3 (0.37) EGFRITGB3ITGAVITGA2BFLT1
SCHEMBL29917902 0.85 ITGB3 (0.37) EGFRITGB3ITGAVITGA2BFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3798214-B1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMA (US) 2022-09-14 EP claimed