SCHEMBL29918436

SCHEMBL29918436

CC(=O)NC(CO)c1cccc(C)c1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 1/20 0.46
HSD17B10 Q99714 1/20 0.45
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RIPK1 Q13546 1/20 0.43
AURKA O14965 1/20 0.42
CDK2 P24941 1/20 0.42
ROCK2 O75116 2/20 0.41
LMNA P02545 1/20 0.41
PAX8 Q06710 1/20 0.41
ACP3 P15309 1/20 0.41
USP1 O94782 1/20 0.40
WDR48 Q8TAF3 1/20 0.40
MAPK1 P28482 2/20 0.40
GPR139 Q6DWJ6 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14393517 1.00 CYP26A1 (0.46) CYP26A1HSD17B10ALDH1A1MAPTL3MBTL1
SCHEMBL4597982 0.89 CYP26A1 (0.50) CYP26A1RIPK1AURKACDK2ROCK2
SCHEMBL23961270 0.86 GPR139 (0.49) CYP26A1HSD17B10RIPK1AURKACDK2
SCHEMBL29675785 0.84 CYP26A1 (0.47) CYP26A1ALDH1A1RIPK1AURKACDK2
SCHEMBL14338245 0.84 KCNA5 (0.46) CYP26A1RIPK1AURKACDK2ROCK2
SCHEMBL18765697 0.84 CYP26A1 (0.47) CYP26A1ALDH1A1RIPK1AURKACDK2
SCHEMBL14393701 0.84 MAPK1 (0.47) PAX8MAPK1
SCHEMBL29751805 0.84 MAPK1 (0.47) PAX8MAPK1
SCHEMBL14393694 0.83 ROCK1 (0.52) CYP26A1ROCK2MAPK1
SCHEMBL14393867 0.83 ROCK1 (0.52) CYP26A1ROCK2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114948963-A Protein kinase inhibitor benzolactam compounds 大冢制药株式会社 2022-08-30 CN disclosed