SCHEMBL29922129

SCHEMBL29922129

O=C1CSc2cc(Br)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.43
PTPRC P08575 1/20 0.38
METAP1 P53582 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.38
BCL2 P10415 2/20 0.37
MCL1 Q07820 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
HSD17B3 P37058 1/20 0.37
PARP10 Q53GL7 2/20 0.37
TDP2 O95551 1/20 0.37
PARP11 Q9NR21 1/20 0.37
HSP90AA1 P07900 1/20 0.34
TLR9 Q9NR96 1/20 0.34
PBRM1 Q86U86 1/20 0.34
KCNN4 O15554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2594793 1.00 S100A4 (0.43) S100A4PTPRCMETAP1KDM4EHTT
SCHEMBL5329304 0.84 S100A4 (0.43) S100A4PTPRCMETAP1BCL2MCL1
SCHEMBL13135 0.81 KDM4E (0.58) S100A4PTPRCMETAP1KDM4EHTT
SCHEMBL5956746 0.78 KDM4E (0.47) S100A4PTPRCMETAP1KDM4EHTT
SCHEMBL6812146 0.76 HTT (0.41) KDM4EHTTCA1CA2CA7
SCHEMBL9159671 0.76 VHL (0.49) S100A4METAP1KDM4EHTTCA1
SCHEMBL13539308 0.76 KDM4E (0.38) KDM4EHTTMAOAMAOB
SCHEMBL13871409 0.76 EPHX2 (0.53) METAP1KDM4EHTTCA1CA2
SCHEMBL31040913 0.73 TDP2 (0.42) KDM4EHTTCA1CA2CA4
SCHEMBL11877796 0.72 MEN1 (0.46) KDM4EHTTPARP10TDP2PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022188735-A1 HETEROCYCLIC COMPOUNDS AS HPK1 INHIBITORS GUANGDONG NEWOPP BIOPHARMACEUTICALS CO., LTD. (CN) 2022-09-15 WO disclosed