SCHEMBL29923628

SCHEMBL29923628

COc1cnc2cccc(N3CCc4ccccc4C3)c2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPK1 P28482 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
NUDT1 P36639 1/20 0.44
GRIN2D O15399 4/20 0.42
GRIN3B O60391 4/20 0.42
GRIN1 Q05586 4/20 0.42
GRIN2A Q12879 4/20 0.42
GRIN2B Q13224 4/20 0.42
GRIN2C Q14957 4/20 0.42
GRIN3A Q8TCU5 4/20 0.42
DRD1 P21728 1/20 0.42
DRD5 P21918 1/20 0.42
CHRM1 P11229 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
LMNA P02545 1/20 0.41
NCF1 P14598 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6159628 0.75 NUDT1 (0.51) MAPTKDM4EMAPK1NPSR1NUDT1
SCHEMBL1223537 0.75 MTNR1B (0.43) MAPTNPSR1NCF1NPC1ALDH1A1
SCHEMBL6159581 0.72 NUDT1 (0.63) MAPTNUDT1GRIN2DGRIN3BGRIN1
Hydrochloric Acid SCHEMBL6162260 0.71 NUDT1 (0.61) MAPTNUDT1GRIN2DGRIN3BGRIN1
SCHEMBL5288680 0.71 PDE10A (0.53) MAPTMAPK1ADRA1DADRA1AADRA1B
SCHEMBL30296979 0.71 DRD1 (0.56) MAPTKDM4EDRD1DRD5LMNA
SCHEMBL27806895 0.71 DRD1 (0.56) MAPTKDM4EDRD1DRD5LMNA
SCHEMBL27946081 0.70 MAPT (0.75) MAPTKDM4EMAPK1NPSR1DRD1
SCHEMBL10536109 0.70 MAPT (0.62) MAPTKDM4EMAPK1NPSR1DRD1
SCHEMBL29978754 0.70 MAPT (0.62) MAPTKDM4EMAPK1NPSR1DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4055013-A1 WDR5 INHIBITORS AND MODULATORS Vanderbilt University (US) 2022-09-14 EP disclosed