SCHEMBL29924345

SCHEMBL29924345

COC(=O)c1ccc2nc(CCl)n(CC3(OC)CC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 1/20 0.44
KDM4E B2RXH2 1/20 0.41
GLP1R P43220 1/20 0.40
DRD2 P14416 2/20 0.40
TBXA2R P21731 2/20 0.40
IDH1 O75874 5/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
OPRK1 P41145 1/20 0.37
CFTR P13569 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29149830 1.00 ACSS2 (0.44) ACSS2KDM4EGLP1RDRD2TBXA2R
SCHEMBL30798065 0.91 ACSS2 (0.42) ACSS2KDM4EGLP1RDRD2TBXA2R
SCHEMBL23363441 0.87 ACSS2 (0.44) ACSS2KDM4EDRD2TBXA2RIDH1
SCHEMBL29664315 0.87 ACSS2 (0.44) ACSS2KDM4EDRD2TBXA2RIDH1
SCHEMBL29555279 0.86 ACSS2 (0.44) ACSS2KDM4EDRD2TBXA2RIDH1
SCHEMBL25340969 0.86 ACSS2 (0.44) ACSS2KDM4EDRD2TBXA2RIDH1
SCHEMBL25340079 0.85 ACSS2 (0.43) ACSS2KDM4EGLP1RDRD2TBXA2R
SCHEMBL29946034 0.85 ACSS2 (0.43) ACSS2KDM4EGLP1RDRD2TBXA2R
SCHEMBL25322110 0.84 ACSS2 (0.42) ACSS2KDM4EDRD2TBXA2RIDH1
SCHEMBL30269530 0.84 ACSS2 (0.42) ACSS2KDM4EDRD2TBXA2RIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed