SCHEMBL29924490

SCHEMBL29924490

O=C(O)c1cc2ncn(C[C@@H]3CCO3)c2s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.37
KDM4E B2RXH2 4/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
TBXAS1 P24557 2/20 0.33
ALDH1A1 P00352 5/20 0.33
RAB9A P51151 1/20 0.33
ABL1 P00519 2/20 0.33
GRIN2B Q13224 1/20 0.32
MAPT P10636 1/20 0.32
BLM P54132 1/20 0.32
TEK Q02763 1/20 0.32
PTGER4 P35408 1/20 0.32
TRPA1 O75762 1/20 0.31
SLC2A1 P11166 1/20 0.31
PLK1 P53350 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30209267 1.00 KDM4C (0.37) KDM4CKDM4EPIK3R1PIK3CATBXAS1
SCHEMBL31025680 0.88 ALDH1A1 (0.37) KDM4EALDH1A1RAB9AABL1SLC2A1
SCHEMBL30209319 0.84 KDM4E (0.37) KDM4CKDM4EPIK3CATBXAS1ALDH1A1
SCHEMBL29924505 0.80 KDM4C (0.37) KDM4CKDM4ETBXAS1ALDH1A1RAB9A
SCHEMBL27143674 0.80 KDM4C (0.37) KDM4CKDM4ETBXAS1ALDH1A1RAB9A
SCHEMBL29586588 0.76 KDM4C (0.38) KDM4CKDM4EALDH1A1GRIN2BMAPT
SCHEMBL30237710 0.75 KDM4C (0.44) KDM4CKDM4EALDH1A1RAB9ATEK
SCHEMBL26611552 0.75 PIK3R1 (0.34) KDM4CKDM4EPIK3R1PIK3CAALDH1A1
SCHEMBL26611555 0.75 PIK3R1 (0.34) KDM4CKDM4EPIK3R1PIK3CAALDH1A1
SCHEMBL23361781 0.72 FGFR1 (0.47) KDM4CGRIN2BPTGER4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed