SCHEMBL29924915

SCHEMBL29924915

Fc1cc2c(Cl)nc(Cl)nc2nc1Cl

nearest known ligand 0.37

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30065127 1.00 KEAP1 (0.37) KEAP1NFE2L2
SCHEMBL24672358 1.00 KEAP1 (0.37) KEAP1NFE2L2
SCHEMBL29795348 0.78 ALDH1A1 (0.30)
SCHEMBL24755330 0.78 ALDH1A1 (0.30)
SCHEMBL2541308 0.72 HTT (0.32) KEAP1NFE2L2
SCHEMBL29909463 0.72 HTT (0.32) KEAP1NFE2L2
SCHEMBL2175712 0.72 GSK3A (0.31)
SCHEMBL31732939 0.71
SCHEMBL29263382 0.71 KEAP1 (0.38) KEAP1NFE2L2
SCHEMBL30577251 0.71 KEAP1 (0.38) KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116375704-A KRAS G12C Preparation and application of mutant protein isoquinolinone inhibitor 药雅科技(上海)有限公司 2023-07-04 CN disclosed
WO-2022193871-A1 PREPARATION AND USE OF KRASG12D MUTANT PROTEIN INHIBITOR 药雅科技(上海)有限公司 2022-09-22 WO disclosed
CN-115073450-A KRAS G12C Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed
CN-115073451-A KRAS G12D Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed