SCHEMBL29930749

SCHEMBL29930749

Nc1cccc(-c2cnc3[nH]ncc3c2)c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIT P10721 6/20 0.55
MAP4K4 O95819 4/20 0.54
NTRK1 P04629 5/20 0.52
PIK3CA P42336 3/20 0.49
ENPP2 Q13822 1/20 0.49
DYRK1A Q13627 1/20 0.48
PIK3C3 Q8NEB9 2/20 0.47
METAP2 P50579 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930718 0.81 AXL (0.61) MAP4K4NTRK1PIK3CADYRK1APIK3C3
SCHEMBL857125 0.79 CDK8 (0.69) KITMAP4K4NTRK1PIK3CADYRK1A
SCHEMBL16914403 0.77 PIK3C3 (0.57) MAP4K4NTRK1PIK3CADYRK1APIK3C3
SCHEMBL8266373 0.75 FGFR1 (0.70) MAP4K4NTRK1DYRK1AMETAP2
SCHEMBL1585618 0.74 CDK8 (0.50) MAP4K4NTRK1PIK3CADYRK1APIK3C3
SCHEMBL978245 0.73 BIRC5 (0.66) KITMAP4K4NTRK1PIK3CA
SCHEMBL22347150 0.73 MAP4K4 (0.49) KITMAP4K4NTRK1ENPP2METAP2
Indazole SCHEMBL28820118 0.73 FGFR1 (0.61) MAP4K4DYRK1AMETAP2
SCHEMBL3376623 0.73 CDK8 (0.73) MAP4K4PIK3C3
SCHEMBL1496196 0.73 MAPT (0.50) MAP4K4NTRK1PIK3CADYRK1APIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed