SCHEMBL29933005

SCHEMBL29933005

NC(=O)c1ccnc(-c2cccc(N3CCOCC3)c2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.62
HDAC1 Q13547 2/20 0.62
KMO O15229 1/20 0.56
PLOD2 O00469 2/20 0.56
PLOD3 O60568 2/20 0.56
PLOD1 Q02809 2/20 0.56
LRRK2 Q5S007 2/20 0.54
STK4 Q13043 1/20 0.54
STK3 Q13188 1/20 0.54
JMJD6 Q6NYC1 1/20 0.53
PIK3R2 O00459 1/20 0.50
ATR Q13535 3/20 0.49
PIK3CA P42336 2/20 0.49
CHEK1 O14757 1/20 0.49
ATRIP Q8WXE1 1/20 0.48
JAK2 O60674 2/20 0.48
CAMK2D Q13557 1/20 0.47
SCN9A Q15858 1/20 0.47
MAPK8 P45983 1/20 0.46
MAPK10 P53779 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29932837 0.88 JAK2 (0.60) KDM1AHDAC1KMOPLOD2PLOD3
SCHEMBL303084 0.84 KMO (0.77) HDAC1KMOPLOD2PLOD3PLOD1
Hydrochloric Acid SCHEMBL14742166 0.83 KMO (0.74) KDM1AHDAC1KMOPLOD2PLOD3
SCHEMBL3722032 0.81 KMO (0.58) KMOPLOD2PLOD3PLOD1LRRK2
SCHEMBL29932887 0.80 KDM1A (0.62) KDM1AHDAC1KMOLRRK2STK4
SCHEMBL3622937 0.79 JAK2 (0.80) HDAC1JAK2CAMK2DMAPK8MAPK10
SCHEMBL27872408 0.76 KDM4B (0.52) KDM1AATR
SCHEMBL3554847 0.75 PIK3CA (0.76) KMOLRRK2STK4STK3ATR
SCHEMBL29889392 0.75 PIK3CA (0.76) KMOLRRK2STK4STK3ATR
SCHEMBL6880915 0.75 LRRK2 (0.52) KMOLRRK2STK4STK3ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113444038-B 2-aryl isonicotinic acid amide LSD1/HDAC double-target inhibitor, and preparation method and application thereof 新乡医学院 2022-09-27 CN disclosed