SCHEMBL29936801

SCHEMBL29936801

OC(c1ccc(OC(F)(F)F)cc1)c1ccc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TOP2A P11388 1/20 0.41
TOP2B Q02880 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
ALDH1A1 P00352 1/20 0.39
IDO1 P14902 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
KDR P35968 1/20 0.38
PDK1 Q15118 1/20 0.38
SLC6A9 P48067 1/20 0.37
NPFFR2 Q9Y5X5 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23388219 1.00 CHEK2 (0.43) CHEK2MEN1KMT2ATOP2ATOP2B
SCHEMBL11441506 0.83 CHEK2 (0.47) CHEK2MEN1KMT2AAKR1C2IDO1
SCHEMBL646362 0.80 TOP2A (0.49) MEN1KMT2ATOP2ATOP2BALDH1A1
SCHEMBL939618 0.77 TOP2A (0.47) MEN1KMT2ATOP2ATOP2BAKR1C2
SCHEMBL23388231 0.77 APLNR (0.43) MEN1KMT2ATOP2ATOP2BAKR1C2
SCHEMBL29936440 0.77 APLNR (0.43) MEN1KMT2ATOP2ATOP2BAKR1C2
SCHEMBL24956326 0.76 HTR3E (0.47) CHEK2PPARGPPARAAKR1C2IDO1
SCHEMBL12782118 0.74 TOP2A (0.44) MEN1KMT2ATOP2ATOP2BAKR1C2
SCHEMBL4603119 0.74 TOP2A (0.51) MEN1KMT2ATOP2ATOP2BALDH1A1
SCHEMBL23388234 0.73 TRPV1 (0.47) CHEK2PPARGPPARAAKR1C2AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4061347-A1 COMPOUNDS FOR USE IN THE TREATMENT OF ACUTE INTERMITTENT PORPHYRIA Vestlandets Innovasjonsselskap AS (NO) 2022-09-28 EP disclosed