SCHEMBL2993822

SCHEMBL2993822

COc1c(Nc2ccccc2)c(=O)c1=O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.51
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
PLK1 P53350 1/20 0.47
CXCR2 P25025 8/20 0.47
MAPT P10636 3/20 0.47
IDO1 P14902 2/20 0.47
MAPK1 P28482 2/20 0.47
MITF O75030 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
BCL9 O00512 1/20 0.47
CTNNB1 P35222 1/20 0.47
HSD17B10 Q99714 2/20 0.42
ALOX12 P18054 1/20 0.42
RAD52 P43351 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2773341 0.90 BCL9 (0.46) POLBMEN1KMT2APLK1CXCR2
SCHEMBL25501940 0.83 CYP1A2 (0.50) POLBMEN1KMT2ACXCR2MAPT
SCHEMBL2773108 0.83 MAPT (0.57) POLBMEN1KMT2AMAPTMAPK1
SCHEMBL2775099 0.81 POLB (0.45) POLBMEN1KMT2ACXCR2MAPT
SCHEMBL2772692 0.81 POLB (0.49) POLBMEN1KMT2ACXCR2MAPT
SCHEMBL2770446 0.81 POLB (0.47) POLBMEN1KMT2ACXCR2MAPT
SCHEMBL2994041 0.81 POLB (0.45) POLBMEN1KMT2AMAPTALDH1A1
SCHEMBL2990917 0.81 KMT2A (0.81) POLBMEN1KMT2AMAPTIDO1
SCHEMBL7785565 0.81 KMT2A (0.60) POLBMEN1KMT2AMAPTMAPK1
SCHEMBL6549773 0.80 POLB (0.68) POLBMEN1KMT2APLK1CXCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240255495-A1 COVALENT APTAMERS UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2024-08-01 US claimed
WO-2022232195-A2 COVALENT APTAMERS UNIVERSITY OF PITTSBURGH-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2022-11-03 WO claimed
US-20260028321-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2026-01-29 US disclosed
CN-120077027-A Sulfonylimide compounds as inhibitors of histone deacetylase 6 and pharmaceutical compositions comprising the same 株式会社钟根堂 2025-05-30 CN disclosed
EP-4504713-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF Chong Kun Dang Pharmaceutical Corp. (KR) 2025-02-12 EP disclosed
CN-119233968-A 1,3, 4-Oxadiazole derivative compounds as histone deacetylase 6 inhibitors and uses thereof 株式会社钟根堂 2024-12-31 CN disclosed
US-20240286994-A1 NOVEL SQUARAMIDE DERIVATIVE AND USE THEREOF PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2024-08-29 US disclosed
US-20240261249-A1 NOVEL SQUARAMIDE DERIVATIVE AND USE THEREOF PUSAN NATIONAL UNIVERSITY INDUSTRY-UNIVERSITY COOPERATION FOUNDATION (KR) 2024-08-08 US disclosed
WO-2023195809-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2023-10-12 WO disclosed
WO-2023195809-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2023-10-12 WO disclosed
CN-112759549-B 3-substituted amino-4- ((substituted pyridinyl) amino) cyclobut-3-ene-1, 2-dione compounds 中国医学科学院药物研究所 2023-07-28 CN disclosed
WO-2022255770-A1 NOVEL SQUARAMIDE DERIVATIVE AND USE THEREOF 부산대학교 산학협력단 2022-12-08 WO disclosed
WO-2021150697-A1 N-SUBSTITUTED-3-TRICYCLYL PIPERIDINE DERIVATIVES AS ANTICANCER AND NEUROPROTECTIVE AGENTS ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2021-07-29 WO disclosed
CN-112759549-A 3-substituted amino-4- ((substituted pyridyl) amino) cyclobut-3-ene-1, 2-diones 中国医学科学院药物研究所 2021-05-07 CN disclosed
US-20100173910-A1 TRIAMINOPYRIMIDINE CYCLOBUTENEDIONE DERIVATIVES USED AS PHOSPHATASE CDC25 INHIBITORS IPDRN PHSTMS D.S.S. (FR) 2010-07-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260028321-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND USES THEREOF HDAC6, HDAC1, HDAC3 POLB 2187/4885MEN1 3823/4885KMT2A 133/4885
US-20100173910-A1 TRIAMINOPYRIMIDINE CYCLOBUTENEDIONE DERIVATIVES USED AS PHOSPHATASE CDC25 INHIBITORS CDC25B, CDC25A, CDC25C POLB 273/4885MEN1 1932/4885KMT2A 1935/4885
US-20240286994-A1 NOVEL SQUARAMIDE DERIVATIVE AND USE THEREOF EIF3E, EIF3A, EIF3K POLB 2038/4885MEN1 3731/4885KMT2A 1471/4885
US-20240261249-A1 NOVEL SQUARAMIDE DERIVATIVE AND USE THEREOF EIF3E, EIF3A, EIF3K POLB 2038/4885MEN1 3731/4885KMT2A 1471/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.