SCHEMBL29939615

SCHEMBL29939615

COCCn1cc(C(N)=O)c(-c2ccccn2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
BTK Q06187 1/20 0.39
MAP4K4 O95819 1/20 0.39
EGFR P00533 1/20 0.39
FRK P42685 1/20 0.39
MAPK9 P45984 1/20 0.39
CSNK1D P48730 1/20 0.39
SLK Q9H2G2 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SMO Q99835 1/20 0.37
PARP1 P09874 1/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30499265 0.83 F12 (0.41) NPSR1RXFP1BTKSMOPARP1
SCHEMBL29725995 0.82 NPSR1 (0.46) NPSR1RXFP1PARP1ALDH1A1IRAK4
SCHEMBL2078208 0.74 IKBKB (0.41) PARP1KDM4EALDH1A1HPGDMAP3K5
SCHEMBL30062375 0.73 MAPT (0.42) L3MBTL1KDM4EALDH1A1RAB9ASMN1; SMN2
Formic Acid SCHEMBL31708378 0.72 TGFBR1 (0.35) MAP4K4EGFRFRKMAPK9CSNK1D
SCHEMBL15048600 0.72 KLK3 (0.47) L3MBTL1KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL20086025 0.71 IRAK4 (0.53) MAP4K4EGFRFRKMAPK9CSNK1D
SCHEMBL19207113 0.70 JMJD6 (0.44) L3MBTL1KDM4EALDH1A1RAB9ASMN1; SMN2
SCHEMBL11606947 0.70 CHEK1 (0.41) NPSR1BTKMAP4K4MAPK9L3MBTL1
SCHEMBL7520947 0.69 PDE10A (0.42) L3MBTL1PARP1KDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110997681-B Thiazolopyridine derivatives as adenosine receptor antagonists 默克专利股份公司 2022-11-15 CN disclosed