SCHEMBL30499265

SCHEMBL30499265

CN(C)CCn1cc(C(N)=O)c(-c2ccccn2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F12 P00748 2/20 0.41
NPSR1 Q6W5P4 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
BTK Q06187 1/20 0.37
KDM5A P29375 1/20 0.37
KDM5B Q9UGL1 1/20 0.37
JAK2 O60674 2/20 0.36
JAK1 P23458 2/20 0.36
JAK3 P52333 2/20 0.36
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
GRM5 P41594 1/20 0.36
CDC7 O00311 1/20 0.36
AURKA O14965 1/20 0.36
NEK2 P51955 1/20 0.36
SMO Q99835 1/20 0.36
ALOX5 P09917 1/20 0.36
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29939615 0.83 NPSR1 (0.40) NPSR1RXFP1BTKJAK2JAK1
SCHEMBL29725995 0.82 NPSR1 (0.46) F12NPSR1RXFP1TGFBR1TGFBR2
SCHEMBL15048610 0.72 PDE10A (0.44) F12NPSR1RXFP1KDM5AKDM5B
SCHEMBL15048614 0.71 PDE10A (0.45) F12KDM5AKDM5BCFTR
SCHEMBL19207113 0.70 JMJD6 (0.44) F12HCRTR1F2
SCHEMBL30839550 0.69 NEK2 (0.49) JAK2JAK1JAK3AURKANEK2
SCHEMBL20577094 0.68 HCRTR1 (0.36) F12KDM5AKDM5BJAK2JAK1
SCHEMBL3620548 0.67 GRM5 (0.51) NPSR1RXFP1TGFBR1TGFBR2GRM5
SCHEMBL23479924 0.67 ADORA1 (0.44) F12NPSR1TGFBR1HCRTR1HCRTR2
SCHEMBL5186668 0.66 TGFBR1 (0.66) TGFBR1TGFBR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096719-A Pyridazinylamino derivatives as ALK5 inhibitors 奇斯药制品公司 2023-05-09 CN disclosed