SCHEMBL29940501

SCHEMBL29940501

COC(=O)c1cc(I)c2ncc(C3CC3)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
PSMD14 O00487 1/20 0.40
ALDH1A1 P00352 3/20 0.38
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
ATM Q13315 1/20 0.36
HSD17B10 Q99714 1/20 0.36
OPRK1 P41145 1/20 0.36
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 2/20 0.34
HPGD P15428 1/20 0.34
AHR P35869 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29278006 1.00 KDM4E (0.41) KDM4EPSMD14ALDH1A1PDGFRBPDGFRA
SCHEMBL21358450 0.86 CYP2C9 (0.40) KDM4EALDH1A1HSD17B10LMNACA12
SCHEMBL23958818 0.85 PDGFRB (0.45) KDM4EPSMD14ALDH1A1PDGFRBPDGFRA
SCHEMBL17442622 0.80 ATM (0.51) KDM4EPSMD14ALDH1A1ATMALOX15
SCHEMBL29940558 0.76 HTT (0.55) KDM4EALDH1A1PDGFRBPDGFRACYP11B1
SCHEMBL19780100 0.76 HTT (0.55) KDM4EALDH1A1PDGFRBPDGFRACYP11B1
SCHEMBL29278003 0.74 ALOX15 (0.39) KDM4EALDH1A1PDGFRBPDGFRAATM
SCHEMBL17067735 0.73 ATM (0.57) KDM4EALDH1A1ATMHSD17B10CYP11B1
SCHEMBL23196216 0.73 PDGFRB (0.46) KDM4EPDGFRBPDGFRAHTTLMNA
SCHEMBL29939947 0.72 HSD17B10 (0.35) KDM4EALDH1A1ATMHSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4308229-A1 INHIBITORS OF PLASMA KALLIKREIN Takeda Pharmaceutical Company Limited (JP) 2024-01-24 EP disclosed
WO-2022197763-A1 INHIBITORS OF PLASMA KALLIKREIN SHIRE HUMAN GENETIC THERAPIES, INC. (US) 2022-09-22 WO disclosed