SCHEMBL29940669

SCHEMBL29940669

CCc1cc2c(cc1C1CCN(C(=O)OC(C)(C)C)CC1)C(C)(C)c1[nH]c3cc(Br)ccc3c1C2

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 6/20 0.48
DPP4 P27487 1/20 0.37
BRD3 Q15059 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
NOTCH1 P46531 4/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
JAK2 O60674 1/20 0.36
FPR2 P25090 2/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27087527 1.00 ALK (0.48) ALKDPP4BRD3KDM4EMAPT
SCHEMBL30009833 0.89 ALK (0.40) ALK
SCHEMBL30009789 0.86 ALK (0.40) ALK
SCHEMBL29940758 0.85 ALK (0.60) ALK
SCHEMBL28913346 0.85 ALK (0.60) ALK
SCHEMBL27087525 0.83 ALK (0.41) ALKPDE4A
SCHEMBL27087547 0.81 ALK (0.36) ALK
SCHEMBL23291507 0.75 MAPT (0.49) DPP4KDM4EMAPTTHRBFPR2
SCHEMBL31222846 0.75 MAPT (0.49) DPP4KDM4EMAPTTHRBFPR2
SCHEMBL31738645 0.74 KDM4E (0.45) DPP4KDM4EMAPTTHRBSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115340523-B Compound with ALK inhibitory activity and preparation method and application thereof 盛世泰科生物医药技术(苏州)股份有限公司 2023-12-15 CN disclosed
CN-115340523-A Compound with ALK inhibitory activity and preparation method and application thereof 盛世泰科生物医药技术(苏州)有限公司 2022-11-15 CN disclosed