SCHEMBL29945202

SCHEMBL29945202

[2H]C([2H])([2H])N1CCC[C@H]1CO[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 5/20 0.43
CHRNA3 P32297 5/20 0.43
CHRNB2 P17787 4/20 0.42
CHRNA4 P43681 3/20 0.42
CHRNA7 P36544 2/20 0.42
CHRNA5 P30532 1/20 0.42
CHRNB1 P11230 2/20 0.40
CHRNB3 Q05901 2/20 0.40
CHRNA1 P02708 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29875863 1.00 CHRNB4 (0.43) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL25906381 0.92 CHRNB2 (0.50) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL22554969 0.82 SMYD2 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL22554967 0.82 SMYD2 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4CHRNA7
SCHEMBL31460034 0.79 SMYD2 (0.38) CHRNB2CHRNA4CHRNA7CHRNA5
SCHEMBL20534267 0.78 FFAR1 (0.46)
SCHEMBL18786265 0.78 FFAR1 (0.46)
SCHEMBL23665772 0.77 CASP3 (0.36) CHRNB2CHRNA4CHRNA7CHRNA5
SCHEMBL31620808 0.76 CASP3 (0.35) CHRNB2CHRNA4CHRNA7CHRNA5
SCHEMBL22554979 0.76 SMYD2 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115073450-A KRAS G12C Preparation and application of mutant protein inhibitor 药雅科技(上海)有限公司 2022-09-20 CN disclosed