SCHEMBL29945825

SCHEMBL29945825

N#Cc1cccc(Br)c1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.41
AR P10275 14/20 0.40
PDK2 Q15119 1/20 0.36
TSHR P16473 1/20 0.34
LMNA P02545 1/20 0.34
PGR P06401 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2134651 1.00 DYRK1A (0.41) DYRK1AARPDK2TSHRLMNA
SCHEMBL25983090 0.85 AR (0.46) ARPDK2TSHRPGR
SCHEMBL21718846 0.80 DYRK1A (0.41) DYRK1AARPDK2TSHRLMNA
SCHEMBL23726465 0.78 HCAR1 (0.40) PDK2TSHRLMNAHCAR1
SCHEMBL1994873 0.78 AR (0.41) ARPDK2TSHRPGR
SCHEMBL3911267 0.78 AR (0.46) ARPGR
SCHEMBL29378798 0.78 AR (0.41) ARPDK2TSHRPGR
SCHEMBL16960191 0.76 AR (0.40) ARPDK2TSHRPGR
SCHEMBL14699104 0.76 DYRK1A (0.42) DYRK1AARPDK2TSHRPGR
SCHEMBL5228912 0.76 TSHR (0.54) ARTSHRPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4663626-A1 IMINE COMPOUNDS AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF Bio Genuine (Shanghai) Biotech Co., Ltd (CN) 2025-12-17 EP disclosed
CN-119546304-A Salts of SOS1 inhibitors 米拉蒂治疗公司 2025-02-28 CN disclosed
CN-119462626-A SOS1 inhibitors 米拉蒂治疗股份有限公司 2025-02-18 CN disclosed
CN-115135315-B SOS1 inhibitors 米拉蒂治疗股份有限公司 2024-11-26 CN disclosed
WO-2024165071-A1 IMINE COMPOUNDS AS WELL AS PREPARATION METHOD THEREFOR AND USE THEREOF 上海葆正医药科技有限公司 2024-08-15 WO disclosed
CN-115135315-A SOS1 inhibitors 米拉蒂治疗股份有限公司 2022-09-30 CN disclosed